| Publication |
Sentence |
Publish Date |
Extraction Date |
Species |
| Manabu Takano, Tsuyoshi Okada, Katsutoshi Shioda, Chikara Yonekawa, Shiro Sud. Risperidone suppresses caffeine-induced hyperthermia and hyperactivity in rats. Neuroscience letters. 2024-09-02. PMID:39222834. |
the rats received intraperitoneal injections of saline, risperidone (0.25 mg/kg, 0.5 mg/kg), way-100635, ketanserin, haloperidol, sulpiride, or sch 23390, 5 min after the administration of caffeine (25 mg/kg). |
2024-09-02 |
2024-09-05 |
rat |
| Olusegun Adebayo Adeoluwa, Anthony Taghogho Eduviere, Gladys Onyinye Adeoluwa, Lily Oghenevovwero Otomewo, Funmilayo Racheal Adeniy. The monoaminergic pathways are involved in the antidepressant-like effect of quercetin. Naunyn-Schmiedeberg's archives of pharmacology. 2023-10-18. PMID:37851059. |
in addition, monoaminergic involvement was investigated by combining quercetin (100 mg/kg) with dopaminergic antagonists (haloperidol and sulpiride), adrenergic blockers (prazosin, propranolol and yohimbine), and serotonergic blockers/inhibitors (metergoline). |
2023-10-18 |
2023-11-08 |
mouse |
| Toshiro Niwa, Yuka Yamamot. Stimulatory and inhibitory effect of antipsychotic agents including dopaminergic neuro-depressants on dopamine formation from p-tyramine mediated by cytochrome P450 2D6. Drug metabolism and bioanalysis letters. 2023-09-15. PMID:37711131. |
the effects of antipsychotic agents, including dopamine d2 receptor blocking agents such as haloperidol, chlorpromazine, and sulpiride, and related compounds such as mirtazapine and sertraline, on dopamine formation from p-tyramine catalyzed by cytochrome p450 (cyp) 2d6.2 (arg296cys;ser486thr), cyp2d6.10 (pro34ser;ser486thr), and cyp2d6.39 (ser486thr) were compared with those of cyp2d6.1. |
2023-09-15 |
2023-10-07 |
Not clear |
| Tuane Bazanella Sampaio, Filipe Neimaier Bilheri, Gilson Rogério Zeni, Cristina Wayne Nogueir. Dopaminergic system contribution to the antidepressant-like effect of 3-phenyl-4-(phenylseleno) isoquinoline in mice. Behavioural brain research. vol 386. 2021-08-24. PMID:32184159. |
lastly, the contribution of dopaminergic system in the psi antidepressant-like effect was demonstrated by using dopamine receptors antagonists, sch23390, haloperidol and sulpiride. |
2021-08-24 |
2023-08-13 |
mouse |
| Vivian M de Vita, Heloisa R Zapparoli, Adriano E Reimer, Marcus L Brandão, Amanda R de Oliveir. Dopamine D2 receptors in the expression and extinction of contextual and cued conditioned fear in rats. Experimental brain research. vol 239. issue 6. 2021-07-28. PMID:33885919. |
to further examine this issue, we evaluated the effects of systemic administration of the dopamine d2-like receptor antagonists sulpiride and haloperidol on the expression and extinction of contextual and cued conditioned fear in rats. |
2021-07-28 |
2023-08-13 |
rat |
| Vivian M de Vita, Heloisa R Zapparoli, Adriano E Reimer, Marcus L Brandão, Amanda R de Oliveir. Dopamine D2 receptors in the expression and extinction of contextual and cued conditioned fear in rats. Experimental brain research. vol 239. issue 6. 2021-07-28. PMID:33885919. |
sulpiride, but not haloperidol, significantly reduced the expression of contextual and cued conditioned fear without affecting extinction recall. |
2021-07-28 |
2023-08-13 |
rat |
| Graziela Vieira, Juliana Cavalli, Elaine C D Gonçalves, Saulo F P Braga, Rafaela S Ferreira, Adair R S Santos, Maíra Cola, Nádia R B Raposo, Raffaele Capasso, Rafael C Dutr. Antidepressant-Like Effect of Terpineol in an Inflammatory Model of Depression: Involvement of the Cannabinoid System and D2 Dopamine Receptor. Biomolecules. vol 10. issue 5. 2021-04-02. PMID:32443870. |
moreover, terpineol showed an antidepressant-like effect in the preventive treatment that was blocked by a nonselective dopaminergic receptor antagonist (haloperidol), a selective dopamine d2 receptor antagonist (sulpiride), a selective cb1 cannabinoid receptor antagonist/inverse agonist (am281), and a potent and selective cb2 cannabinoid receptor inverse agonist (am630), but it was not blocked by a nonselective adenosine receptor antagonist (caffeine) or a β-adrenoceptor antagonist (propranolol). |
2021-04-02 |
2023-08-13 |
Not clear |
| M. Yamaguchi, K. Kimura-Iwasaki, T. Akai, Y. Nakada, H. Nakagaw. Terguride, a dopamine D(2) partial agonist, as a discriminative stimulus in rats. Behavioural pharmacology. vol 2. issue 3. 2019-11-20. PMID:11224067. |
the d(1) agonist skf38393, the da antagonist haloperidol, the d(2) antagonist sulpiride, the d(1) antagonist sch23390, the 5-ht(1a) agonist 8-oh-dpat, the 5-ht(1b) agonist m-cpp and the 5-ht(2) agonist doi were not generalized. |
2019-11-20 |
2023-08-12 |
rat |
| L.E. Baker, E.E. Riddle, R.B. Saunders, J.B. Appe. The role of monoamine uptake in the discriminative stimulus effects of cocaine and related compounds. Behavioural pharmacology. vol 4. issue 1. 2019-11-20. PMID:11224173. |
when given in combination with cocaine, cis flupenthixol and sch 23390 reduced responding on the cocaine-appropriate lever significantly and to a greater extent than either haloperidol, (+/-) sulpiride or (-) sulpiride; neither (+) sulpiride nor metergoline had significant effects. |
2019-11-20 |
2023-08-12 |
rat |
| D. Fontana, R.M. Post, S.R.B. Weiss, A. Per. The role of D1 and D2 dopamine receptors in the acquisition and expression of cocaine-induced conditioned increases in locomotor behavior. Behavioural pharmacology. vol 4. issue 4. 2019-11-20. PMID:11224206. |
pretreatment with d1 (sch 23390) or d2 (raclopride, sulpiride, haloperidol) da antagonists on day 1 prevented the development of conditioning as assessed on day 2, indicating that both receptor subtypes are involved in acquisition. |
2019-11-20 |
2023-08-12 |
rat |
| Jocelyne Caboche, Philippe Vernier, Monique Rogard, Jean-François Julien, Jacques Mallet, Marie-Jo Besso. Role of Dopaminergic D2 Receptors in the Regulation of Glutamic Acid Decarboxylase Messenger RNA in the Striatum of the Rat. The European journal of neuroscience. vol 4. issue 5. 2019-11-20. PMID:12106353. |
levels of messenger rna (mrna) encoding glutamic acid decarboxylase (gad) and preproenkephalin (ppe) were measured by northern blot and in situ hybridization analyses in the striatum of the rat, after chronic injections of two neuroleptics, sulpiride and haloperidol. |
2019-11-20 |
2023-08-12 |
rat |
| Behzad Mesbahzadeh, Nasroallah Moradi-Kor, Saeid Abbasi-Malek. Zinc enhances the expression of morphine-induced conditioned place preference through dopaminergic and serotonergic systems. Biomolecular concepts. vol 10. issue 1. 2019-11-20. PMID:30956225. |
pre-treatment with dopamine receptor antagonists (sch23390, sulpiride, and haloperidol) and serotonin receptor antagonists (way100135, ketanserin, and ondansetron) reversed the enhancement effect of zn on the expression of morphine-induced cpp (especially 20mg/kg, i.p. |
2019-11-20 |
2023-08-13 |
rat |
| Hung-Yu Chan, Yi-Ju Pan, Jiahn-Jyh Chen, Chiung-Hsu Che. Time to Discontinuation of Second-Generation Antipsychotics Versus Haloperidol and Sulpiride in People With Schizophrenia: A Naturalistic, Comparative Study. Journal of clinical psychopharmacology. vol 37. issue 1. 2017-06-05. PMID:27977467. |
time to discontinuation of second-generation antipsychotics versus haloperidol and sulpiride in people with schizophrenia: a naturalistic, comparative study. |
2017-06-05 |
2023-08-13 |
Not clear |
| Berenice Venegas-Meneses, José Francisco Padilla, Claudia Elvira Juárez, José Luis Morán, Carolina Morán, Nora Hilda Rosas-Murrieta, Anabella Handal, Roberto Domíngue. Effects of ovarian dopaminergic receptors on ovulation. Endocrine. vol 50. issue 3. 2016-09-26. PMID:26024972. |
the following treatments blocked ovulation: injecting haloperidol to rats on estrus or diestrus-1 at 8:00, 13:00, or 20:00 h and to rats on diestrus-2 at 08:00, or 20:00 h; injecting sch-23390 to rats on diestrus-1 at 8:00, 13:00, or 20:00 h; injecting sulpiride to rats on estrus at 20:00 h, diestrus-1 at 08:00, 13:00, or 20:00 h and to rats on diestrus-2 at 08:00 h. in rats treated with any of the dopamine antagonists that blocked ovulation, injecting gnrh at 14.00 h on the next predicted proestrus day restored ovulation. |
2016-09-26 |
2023-08-13 |
rat |
| Alessandro Tomassini, Diane Ruge, Joseph M Galea, William Penny, Sven Bestman. The Role of Dopamine in Temporal Uncertainty. Journal of cognitive neuroscience. vol 28. issue 1. 2016-09-15. PMID:26401816. |
in a placebo-controlled double-blind design using a selective d2-receptor antagonist (sulpiride) and d1/d2 receptor antagonist (haloperidol), participants performed a variable foreperiod reaching task, under different conditions of internal and external temporal uncertainty. |
2016-09-15 |
2023-08-13 |
human |
| Małgorzata Hołuj, Piotr Popik, Agnieszka Nikiforu. Improvement of ketamine-induced social withdrawal in rats: the role of 5-HT7 receptors. Behavioural pharmacology. vol 26. issue 8 Spec No. 2016-08-22. PMID:25769091. |
acute administration of amisulpride (3 mg/kg) and sb-269970 (1 mg/kg), a 5-ht7 receptor antagonist, reversed ketamine-induced social withdrawal, whereas sulpiride (20 or 30 mg/kg) and haloperidol (0.2 mg/kg) were ineffective. |
2016-08-22 |
2023-08-13 |
rat |
| Kensuke Sakuma, Hidetoshi Komatsu, Minoru Maruyama, Sachiko Imaichi, Yugo Habata, Masaaki Mor. Temporal and spatial transcriptional fingerprints by antipsychotic or propsychotic drugs in mouse brain. PloS one. vol 10. issue 2. 2015-12-01. PMID:25693194. |
our data showed that various types of antipsychotics with a profound interaction of d2r including haloperidol (antagonist), olanzapine (antagonist), and aripiprazole (partial agonist) all share common spatial tfps closely homologous to those of d2r antagonist sulpiride, and elicited greater transcriptional responses in the striatum than in the nucleus accumbens. |
2015-12-01 |
2023-08-13 |
mouse |
| Timothy J Donahue, Todd M Hillhouse, Kevin A Webster, Richard Young, Eliseu O De Oliveira, Joseph H Porte. (S)-amisulpride as a discriminative stimulus in C57BL/6 mice and its comparison to the stimulus effects of typical and atypical antipsychotics. European journal of pharmacology. vol 734. 2015-01-28. PMID:24726559. |
in tests of stimulus generalization, the (s)-amisulpride stimulus generalized completely to sulpiride (ed50=12.67mg/kg; 37.1µmol/kg), a benzamide analog that also is purported to be an atypical antipsychotic, but did not fully generalize to the typical antipsychotic drug haloperidol (maximum of 45% drug-lever responding) nor to the atypical antipsychotic drugs clozapine (partial substitution of 65% drug-lever responding) or aripiprazole (~30% drug-lever responding). |
2015-01-28 |
2023-08-13 |
mouse |
| L E B Savio, F C Vuaden, L W Kist, T C Pereira, D B Rosemberg, M R Bogo, C D Bonan, A T S Wys. Proline-induced changes in acetylcholinesterase activity and gene expression in zebrafish brain: reversal by antipsychotic drugs. Neuroscience. vol 250. 2014-04-04. PMID:23867765. |
moreover, the proline-induced increase on ache activity was completely reverted by acute administration of antipsychotic drugs (haloperidol and sulpiride), as well as the changes induced in ache expression. |
2014-04-04 |
2023-08-12 |
zebrafish |
| Edward Chia-Cheng Lai, Chia-Hsien Chang, Yea-Huei Kao Yang, Swu-Jane Lin, Chia-Yin Li. Effectiveness of sulpiride in adult patients with schizophrenia. Schizophrenia bulletin. vol 39. issue 3. 2013-10-28. PMID:22315480. |
after adjusting for patient demographics, mental illness characteristics, and propensity score, the cox regression models found that the risk of nonpersistence was significantly higher in patients receiving risperidone (hazard ratio [hr], 1.22; 95% ci, 1.06-1.40), haloperidol (hr, 1.98; 95% ci, 1.63-2.40), and olanzapine (hr, 1.34; 95% ci, 1.07-1.68), as compared with sulpiride, suggesting the effectiveness of sulpiride was better than the other 3 antipsychotics. |
2013-10-28 |
2023-08-12 |
Not clear |